Synthesis and antimicrobial activity of some pyrazoline derivatives bearing amide moiety

Year 2013, Volume: 17 Issue: 3, 187 - 192, 07.03.2014

Ahmet Özdemir

Abstract

Keywords

pyrazoline, amide, furan, thiophene, antimicrobial activity

References

• Alanis AJ. Resistance to antibiotics: Are we in the postantibiotic era?. Arch Med Res 2005; 36: 697-705.
• Ghannoum MA, Louis BR. Antifungal agents: mode of action, mechanisms of resistance and correlation of these mechanisms with bacterial resistance. Clin Microbiol Rev 1999; 12: 501-17.
• Palkar M, Noolvi M, Sankangoud R, Maddi V, Gadad A, Nargund LVG. Synthesis and antibacterial activity of a novel series of 2,3-diaryl-substituted-imidazo(2,1-b)benzothiazole derivatives. Arch Pharm Chem Life Sci 2010; 343: 353-9.
• Lemke TL, Williams DA. Foye’s Principles of Medicinal Chemistry. Lippincott Williams&Wilkins, Baltimore and Philadelphia. 2008.
• Papich MG, Riviere JE. Veterinary pharmacology and therapeutics. Wiley-Blackwell, Iowa. 2009.
• Ciapetti P, Giethlen B. The Practice of Medicinal Chemistry. Academic Press, Burlington. 2008.
• Lima LM, Barreiro EJ. Bioisosterism: A useful strategy for molecular modification and drug design. Curr Med Chem 2005; 12: 23-49.
• Patani GA, LaVoie EJ. Bioisosterism: A rational approach in drug design. Chem Rev 1996; 96: 3147-76.
• Narang R, Narasimhan B, Sharma S. A review on biological activities and chemical synthesis of hydrazide derivatives. Curr Med Chem 2012; 19: 569-612.
• Suresh K, Sandhya B, Sushma D, Rajiv K, Himanshu G. Biological activities of pyrazoline derivatives - A recent development. Recent Patents Anti-Infect Drug Discov 2009; 4: 154-63.
• Kaplancıklı ZA, Turan-Zitouni G, Özdemir A, Revial G, Güven K. Synthesis and antimicrobial activity of some thiazolyl-pyrazoline derivatives. Phosphorus Sulfur Silicon Relat Elem 2007; 182: 749-64.
• Özdemir A, Turan-Zitouni G, Kaplancıklı ZA, Revial G, Güven K. Synthesis and antimicrobial activity of 1-(4-aryl-2-thiazolyl)-3-(2-thienyl)-5-aryl-2-pyrazoline derivatives. Eur J Med Chem 2007; 42: 403-9.
• Özdemir A, Turan-Zitouni G, Kaplancıklı ZA, Revial G, Demirci F, Iscan G. Preparation of some pyrazoline derivatives and evaluation of their antifungal activities. J Enzym Inhib Med Chem 2010; 25: 565-71.
• Turan-Zitouni G, Özdemir A, Güven K. Synthesis of some 1-[(N,Ndisubstituted thiocarbamoylthio)acetyl]3-(2-thienyl)-5-aryl-2-pyrazoline derivatives and investigation of their antibacterial and antifungal activities. Arch Pharm Pharm Med Chem 2005; 338: 96-104.
• Turan-Zitouni G, Özdemir A, Kaplancıklı ZA. Synthesis and antimicrobial activities of some 1-[(N,N-disubstitutedthiocarbamoylthio)acetyl]-3,5-diaryl-2-pyrazolines. Phosphorus Sulfur Silicon Relat Elem 2005; 180: 2717-24.
• Kabli RA, Khalaf AA, Zimaity MT, Khalil AM, Kaddah AM, Al-Rifaie HA. Synthesis of a new series of furyl and thienyl substituted pyrazolines starting with furyl and thienyl chalcones. J Indian Chem Soc 1991; 68: 47-51.
• Khalaf AA, Kabli RA, Zimaity MT, Khalil AM, Kaddah AM, Al-Rifaie, HA. N-Derivatization of some 3-(2-furyl)and 3-(2-thienyl)-5-aryl-2-pyrazolines. Indian J Chem Sect B 1993; 32: 1125-9.
• Winn WC, Allen SD, Janda WM, Koneman EW, Procop GW, Schreckenberger PC, Woods GL. Koneman’s color atlas and textbook of diagnostic microbiology. Lippincott Williams&Wilkins, Baltimore and Philadelphia. 200 Ledneczki I, Forgo P, Kiss JT, Molnár Á, Pálinkó I. Conformational behaviour of acetamide derivatives studied by NMR spectroscopic and computational methods. J Mol Struct 2007; 834: 349-54.
• Vijayabaskar V, Perumal S, Selvaraj S, Lycka A, Murugan R, Balasubramanian M. Synthesis and multinuclear NMR study of (E)-s-trans-1-acetyl-5-aryl-3-styryl2-pyrazolines. Magn Reson Chem 1999; 37: 133-9.